What Is IGF-1?

IGF-1 (Insulin-like Growth Factor 1, also called Somatomedin C) is a 70-amino acid peptide hormone structurally similar to insulin. It's primarily produced by the liver in response to growth hormone (GH) stimulation and mediates many of GH's anabolic effects on tissues throughout the body.

Amino Acids: 70 Molecular Weight: 7,649 Da Production: Liver (mainly), also local tissue synthesis Regulation: GH-dependent and GH-independent Clinical Product: Mecasermin (Increlex®)

Key Characteristics

  • Role: Primary mediator of growth hormone effects
  • Structure: Similar to insulin (hence "insulin-like")
  • Binding: Circulates bound to IGFBPs (binding proteins)
  • Effects: Growth, anabolic, anti-apoptotic

GH → IGF-1 Axis

Understanding the GH/IGF-1 relationship:

  • GH stimulates liver to produce IGF-1
  • IGF-1 provides negative feedback on GH release
  • Many GH effects are mediated through IGF-1
  • Some GH effects are direct (not IGF-1 dependent)
  • IGF-1 is used clinically as marker of GH status

Biological Functions

  • Growth: Essential for linear growth in children
  • Anabolic: Protein synthesis in muscle
  • Metabolic: Glucose uptake, fat metabolism
  • Cell survival: Anti-apoptotic effects
  • Brain: Neurogenesis and neuroprotection

Clinical Use

Mecasermin (recombinant IGF-1) is FDA-approved for:

  • Primary IGF-1 deficiency (GH insensitivity)
  • Laron syndrome (GH receptor defect)
  • GH gene deletion with antibodies to GH

Variants and Analogs

CompoundDescriptionNotes
IGF-1Native 70 aaShort half-life
IGF-1 LR383 aa, modifiedResearch; longer half-life
IGF-1 DES67 aa, truncatedResearch; more potent locally
MGFMechano-Growth FactorIGF-1 splice variant

IGF-1 and Aging/Longevity

Interestingly, the IGF-1/longevity relationship is complex:

  • Low IGF-1 associated with extended lifespan in some species
  • Laron syndrome patients (no IGF-1) have low cancer rates
  • High IGF-1 may increase certain cancer risks
  • The "growth-longevity tradeoff" concept

Medical Use Only

IGF-1 (Mecasermin) is a prescription medication with significant side effects including hypoglycemia, increased intracranial pressure, and potential cancer risk concerns. Research forms like IGF-1 LR3 are not approved for human use. IGF-1 use is banned in sports.

Summary

IGF-1 is the key downstream mediator of growth hormone's effects on tissues. While essential for normal growth and development, it also raises interesting questions about the tradeoff between growth/anabolism and longevity. Clinical use is limited to specific deficiency states due to side effect concerns.

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